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Mostrati risultati da 21 a 40 di 46
Titolo Anno di pubblicazione Autori Unitn File
Cell-permeable dual inhibitors of protein kinases CK2 and PIM-1: Structural features and pharmacological potential 1-gen-2014 Lolli, Graziano +
Active Form of the Protein Kinase CK2 alpha(2)beta(2) holoenzyme Is a Strong Complex with Symmetric Architecture 1-gen-2014 LOLLI, GRAZIANO +
Structural characterization of the STAS domain of prestin. 1-gen-2015 Lolli, Graziano +
Structural Basis of CK2 Regulation by Autoinhibitory Oligomerization 1-gen-2015 Lolli, Graziano +
The "gatekeeper" Residue Influences the Mode of Binding of Acetyl Indoles to Bromodomains 1-gen-2016 Lolli, Graziano +
High-Throughput Fragment Docking into the BAZ2B Bromodomain: Efficient in Silico Screening for X-Ray Crystallography 1-gen-2016 Lolli, Graziano +
The STAS domain of mammalian SLC26A5 prestin harbours an anion-binding site 1-gen-2016 Lolli, Graziano +
Derivatives of 3-Amino-2-methylpyridine as BAZ2B Bromodomain Ligands: In Silico Discovery and in Crystallo Validation 1-gen-2016 Lolli, Graziano +
Characterization of the oligomeric states of the CK2 α2β2 holoenzyme in solution 1-gen-2017 Lolli, Graziano +
Discovery of BAZ2A bromodomain ligands 1-gen-2017 Lolli, Graziano +
Discovery of Inhibitors of Four Bromodomains by Fragment-Anchored Ligand Docking 1-gen-2017 Dalle Vedove, AndreaLolli, Graziano +
Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains 1-gen-2018 Dalle Vedove A.D'Agostino V. G.Lolli G. +
Insight into GFPmut2 pH Dependence by Single Crystal Microspectrophotometry and X-ray Crystallography 1-gen-2018 Lolli, Graziano +
Screening Approaches for Targeting Ribonucleoprotein Complexes: A New Dimension for Drug Discovery 1-gen-2019 D’Agostino, Vito GiuseppeSighel, DeniseZucal, ChiaraBonomo, IsabelleMicaelli, MariachiaraLolli, GrazianoProvenzani, AlessandroQuattrone, AlessandroAdami, Valentina
Inhibitory Properties of ATP-Competitive Coumestrol and Boldine Are Correlated to Different Modulations of CK2 Flexibility 1-gen-2019 Lolli G. +
Biochemical and cellular mechanism of protein kinase CK2 inhibition by deceptive curcumin 1-gen-2020 Dalle Vedove A.Lolli G. +
A novel class of selective CK2 inhibitors targeting its open hinge conformation 1-gen-2020 Dalle Vedove A.Zonta F.Cazzanelli G.Lolli G. +
Identification of compounds inhibiting prion replication and toxicity by removing PrPC from the cell surface 1-gen-2020 Biggi S.Pancher M.Stincardini C.Massignan T.Dalle Vedove A.Gatto P.Lolli G.Adami V.Biasini E. +
Identification of a BAZ2A Bromodomain Hit Compound by Fragment Joining 1-gen-2021 Dalle Vedove, AndreaCazzanelli, GiuliaCorsi, JessicaD’Agostino, Vito GiuseppeLolli, Graziano +
Pharmacological inactivation of the prion protein by targeting a folding intermediate 1-gen-2021 Spagnolli, GiovanniMassignan, TaniaBiggi, SilviaRigoli, MartaLibergoli, MichelaIaneselli, AlanOrioli, SimoneBoldrini, AlbertoBonaldo, ValerioMaietta, GiuliaTosatto, LauraVignoli, BeatricePetris, GianlucaPennuto, MariaGuella, GrazianoCanossa, MarcoLolli, GrazianoBiressi, StefanoMancini, InesFaccioli, PietroBiasini, Emiliano +
Mostrati risultati da 21 a 40 di 46
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