Sfoglia per Autore
Cell-permeable dual inhibitors of protein kinases CK2 and PIM-1: Structural features and pharmacological potential
2014-01-01 Cozza, Giorgio; Girardi, Cristina; Ranchio, Alessandro; Lolli, Graziano; Sarno, Stefania; Orzeszko, Andrzej; Kazimierczuk, Zygmunt; Battistutta, Roberto; Ruzzene, Maria; Pinna, Lorenzo A.
Active Form of the Protein Kinase CK2 alpha(2)beta(2) holoenzyme Is a Strong Complex with Symmetric Architecture
2014-01-01 Lolli, Graziano; Ranchio, Alessandro; Battistutta, Roberto
Structural characterization of the STAS domain of prestin.
2015-01-01 Costanzi, Elisa; Lolli, Graziano; Pasqualetto, Elisa; Bonetto, Greta; Battistutta, Roberto
Structural Basis of CK2 Regulation by Autoinhibitory Oligomerization
2015-01-01 Lolli, Graziano; Battistutta, Roberto
The "gatekeeper" Residue Influences the Mode of Binding of Acetyl Indoles to Bromodomains
2016-01-01 Unzue, Andrea; Zhao, Hongtao; Lolli, Graziano; Dong, Jing; Zhu, Jian; Zechner, Melanie; Dolbois, Aymeric; Caflisch, Amedeo; Nevado, Cristina
High-Throughput Fragment Docking into the BAZ2B Bromodomain: Efficient in Silico Screening for X-Ray Crystallography
2016-01-01 Lolli, Graziano; Caflisch, Amedeo
The STAS domain of mammalian SLC26A5 prestin harbours an anion-binding site
2016-01-01 Lolli, Graziano; Pasqualetto, Elisa; Costanzi, Elisa; Bonetto, Greta; Battistutta, Roberto
Derivatives of 3-Amino-2-methylpyridine as BAZ2B Bromodomain Ligands: In Silico Discovery and in Crystallo Validation
2016-01-01 Marchand, Jean Rémy; Lolli, Graziano; Caflisch, Amedeo
Characterization of the oligomeric states of the CK2 α2β2 holoenzyme in solution
2017-01-01 Lolli, Graziano; Naressi, Denise; Sarno, Stefania; Battistutta, Roberto
Discovery of BAZ2A bromodomain ligands
2017-01-01 Spiliotopoulos, Dimitrios; Wamhoff, Eike-christian; Lolli, Graziano; Rademacher, Christoph; Caflisch, Amedeo
Discovery of Inhibitors of Four Bromodomains by Fragment-Anchored Ligand Docking
2017-01-01 Marchand, Jean-Rémy; Dalle Vedove, Andrea; Lolli, Graziano; Caflisch, Amedeo
Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains
2018-01-01 Dalle Vedove, A.; Spiliotopoulos, D.; D'Agostino, V. G.; Marchand, J. -R.; Unzue, A.; Nevado, C.; Lolli, G.; Caflisch, A.
Insight into GFPmut2 pH Dependence by Single Crystal Microspectrophotometry and X-ray Crystallography
2018-01-01 Lolli, Graziano; Raboni, Samanta; Pasqualetto, Elisa; Benoni, Roberto; Campanini, Barbara; Ronda, Luca; Mozzarelli, Andrea; Bettati, Stefano; Battistutta, Roberto
Screening Approaches for Targeting Ribonucleoprotein Complexes: A New Dimension for Drug Discovery
2019-01-01 D’Agostino, Vito Giuseppe; Sighel, Denise; Zucal, Chiara; Bonomo, Isabelle; Micaelli, Mariachiara; Lolli, Graziano; Provenzani, Alessandro; Quattrone, Alessandro; Adami, Valentina
Inhibitory Properties of ATP-Competitive Coumestrol and Boldine Are Correlated to Different Modulations of CK2 Flexibility
2019-01-01 Battistutta, R.; Lolli, G.
Biochemical and cellular mechanism of protein kinase CK2 inhibition by deceptive curcumin
2020-01-01 Cozza, G.; Zonta, F.; Dalle Vedove, A.; Venerando, A.; Dall'Acqua, S.; Battistutta, R.; Ruzzene, M.; Lolli, G.
A novel class of selective CK2 inhibitors targeting its open hinge conformation
2020-01-01 Dalle Vedove, A.; Zonta, F.; Zanforlin, E.; Demitri, N.; Ribaudo, G.; Cazzanelli, G.; Ongaro, A.; Sarno, S.; Zagotto, G.; Battistutta, R.; Ruzzene, M.; Lolli, G.
Identification of compounds inhibiting prion replication and toxicity by removing PrPC from the cell surface
2020-01-01 Biggi, S.; Pancher, M.; Stincardini, C.; Luotti, S.; Massignan, T.; Dalle Vedove, A.; Astolfi, A.; Gatto, P.; Lolli, G.; Barreca, M. L.; Bonetto, V.; Adami, V.; Biasini, E.
Identification of a BAZ2A Bromodomain Hit Compound by Fragment Joining
2021-01-01 Dalle Vedove, Andrea; Cazzanelli, Giulia; Corsi, Jessica; Sedykh, Maria; D’Agostino, Vito Giuseppe; Caflisch, Amedeo; Lolli, Graziano
Pharmacological inactivation of the prion protein by targeting a folding intermediate
2021-01-01 Spagnolli, Giovanni; Massignan, Tania; Astolfi, Andrea; Biggi, Silvia; Rigoli, Marta; Brunelli, Paolo; Libergoli, Michela; Ianeselli, Alan; Orioli, Simone; Boldrini, Alberto; Terruzzi, Luca; Bonaldo, Valerio; Maietta, Giulia; Lorenzo, Nuria L; Fernandez, Leticia C; Codeseira, Yaiza B; Tosatto, Laura; Linsenmeier, Luise; Vignoli, Beatrice; Petris, Gianluca; Gasparotto, Dino; Pennuto, Maria; Guella, Graziano; Canossa, Marco; Altmeppen, Hermann C; Lolli, Graziano; Biressi, Stefano; Pastor, Manuel M; Requena, Jesús R; Mancini, Ines; Barreca, Maria L; Faccioli, Pietro; Biasini, Emiliano
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